Exemestanex – 20mg/tab

Description

Exemestane, marketed under the brand name Aromasin, was originally developed in the late 1990s as a potential treatment for cancer. Following successful clinical trials that showed its superiority over Tamoxifen, Pfizer released Aromasin to the market. This medication has since become a popular choice in the bodybuilding community, as its effectiveness in reducing estrogen levels has been well-documented. Aromasin is now widely included in underground lab product offerings worldwide.

Aromasin is classified as a Suicidal Aromatase Inhibitor and is typically administered orally. Its primary use is to help regulate estrogen levels in the body, which is crucial for preventing estrogenic side effects and maintaining a lean and dry physique, especially during competitions. Aromasin achieves this by binding to the aromatase enzyme, which is responsible for converting testosterone and other aromatizable drugs into estrogen. By permanently deactivating the aromatase enzyme, Aromasin prevents estrogen rebound, distinguishing it from other anti-estrogens.

Unlike some other aromatase inhibitors, Aromasin requires frequent dosing to maintain optimal levels in the body, ideally every 12 hours. This frequent dosing schedule sets Aromasin apart from other AI’s that can be taken less frequently. Additionally, Aromasin has been shown to have a neutral impact on cholesterol levels, making it a safer option for heart health compared to other anti-estrogens.

In conclusion, Aromasin’s unique mechanism of action and favorable safety profile make it a preferred choice for bodybuilders and individuals seeking to manage estrogen levels effectively. Its ability to maintain a hard and dry appearance without compromising heart health sets it apart as a valuable tool in the world of performance enhancement.

Exemestane is a synthetic androgen analogue that acts as a steroidal inhibitor of aromatase. This medication binds irreversibly to and inhibits the enzyme aromatase, preventing the conversion of cholesterol to pregnenolone and the peripheral aromatization of androgen precursors into estrogens. While Exemestane has been associated with a low rate of serum enzyme elevations during therapy and rare instances of clinically apparent liver injury, it is primarily used to treat certain types of cancer, such as hormone-receptor-positive cancer, in postmenopausal women.

Additionally, Exemestane is utilized to help prevent the recurrence of cancer. Some cancers are fueled by the natural hormone estrogen, and Exemestane works by reducing the body’s production of estrogen, thereby slowing or reversing the growth of these cancers. It is important to note that Exemestane is typically not prescribed for women of childbearing age.

The recommended dosage of Exemestane is once a day after a meal, taken at the same time each day. Treatment with Exemestane may be necessary for several years or longer, and it is crucial to continue taking the medication even if you are feeling well. It is imperative to consult with your doctor before discontinuing the use of Exemestane.

Anabolic-Androgenic Ratio: Not applicable.
Aromatizable: No. It exhibits anti-estrogenic activity.
Progestagenic Activity: None.
Methylated: No.

Standard Dosing Range and Cycle Length: Aromasin is commonly prescribed at a dosage of 12.5-50 mg per day. The specific dosing requirements will be determined based on the number, type, and amount of aromatizable drugs being used. Aromasin is typically administered for as long as aromatizable drugs are being used.

Frequency of Administration: Aromasin should be taken daily, split into 2 equally divided doses.